In:
European Journal of Organic Chemistry, Wiley, Vol. 2015, No. 17 ( 2015-06), p. 3743-3750
Abstract:
An effective and practical palladium‐catalyzed C2‐acylation method was successfully developed for the synthesis of 2‐acylindoles. A variety of 2‐acylindoles were readily prepared from N ‐pyrimidyl indoles in moderate to good yields. This methodology offers several advantages, which include ease of handling, mild reaction conditions, and use of an efficient and cheap catalyst. In particular, challenging 2‐acetylindoles were synthesized in good yields.
Type of Medium:
Online Resource
ISSN:
1434-193X
,
1099-0690
DOI:
10.1002/ejoc.v2015.17
DOI:
10.1002/ejoc.201500304
Language:
English
Publisher:
Wiley
Publication Date:
2015
detail.hit.zdb_id:
1475010-7
Permalink